Tianeptine Metabolite MC5-d4 is an opioid substance, an active metabolite of tianeptine (also called Stablon, Tatinol, Coaxil), a substance developed for the treatment of depression, anxiety, irritable bowel treatment, asthma.
Chemistry
Tianeptine Metabolite MC5-d4 has a similar chemical structure to tianeptine.
Pharmacology
This substance is relatively new and there is little data on its toxicological and pharmacological properties.
Studies in mice have shown that this substance acts as an atypical agonist of the μ-opioid receptors with a clinically insignificant effect on the δ- and κ-opioid receptors. It can cause a calming effect on the body, has a beneficial effect on cognitive abilities, acts as a selective serotonin reuptake inhibitor, serotonin and norepinephrine reuptake inhibitor.
Legal status
Tianeptine Metabolite MC5-d4 may be controlled by law in those countries where Tianeptine and its analogues are controlled substances.
Product Name: Tianeptine Metabolite MC5-d4
Other Name(s):
IUPAC Name: sodium;5-[(3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]benzothiazepin-11-yl)amino]-3,3,4,4-tetradeuteriopentanoate;
7-[(3-Chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepin-11-yl)amino]pentanoic Acid S,S-Dioxide-d4 Sodium Salt;
CAS: 1330171-36-2, 115220-11-6
Molar Mass: 434.9
Molecular Formula: C19H20ClN2NaO4S
InChi Code: InChI=1S/C19H21ClN2O4S.Na/c1-22-16-7-3-2-6-14(16)19(21-11-5-4-8-18(23)24)15-10-9-13(20)12-17(15)27(22,25)26;/h2-3,6-7,9-10,12,19,21H,4-5,8,11H2,1H3,(H,23,24);/q;+1/p-1/i4D2,5D2;
InChIKey: GBYSEZGRQUELJJ-HGFPCDIYSA-M
Canonical SMILES: CN1C2=CC=CC=C2C(C3=C(S1(=O)=O)C=C(C=C3)Cl)NCCCCC(=O)[O-].[Na+]
Formulation: A solid
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